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日期：2023-02-16 作者: . 来源：生命科学与健康工程学院

2022年
序号	论文名称	来源期刊	收录情况
1	Highly efficient decontamination of tetracycline and pathogen by a natural product-derived Emodin/HAp photocatalyst	Chemosphere	SCI
2	Efficient synthesis of rebaudioside D2 through UGT94D1-catalyzed regio-selective glycosylation	Carbohydrate Research	SCI
3	Synthesis and biological evaluation of new series of quinazoline derivatives as EGFR/HER2 dual-target inhibitors	Bioorganic & Medicinal Chemistry Letters	SCI
4	Synthesis and biological evaluation of novel 5,6-dihydrobenzo[h]quinazoline derivatives as FLT3 inhibitors	Chemical Biology & Drug Design	SCI
5	Pyrizolo[1,5-a]pyrimidine derivatives of the second-generation TRK inhibitor: Design, synthesis and biological evaluation	Bioorganic & Medicinal Chemistry Letters	SCI

2021年
序号	论文名称	来源期刊	收录情况
1	Discovery and Validation of a Novel Target of Molluscicides against Oncomelania hupensis, the Intermediate Host of Schistosoma japonicum	Acta Tropica	SCI
2	Evaluation of the molluscicidal activities of arylpyrrole on Oncomelania hupensis, the intermediate host of Schistosoma japonicum	PeerJ	SCI
3	Pyrazolo[1,5-a]pyrimidine based Trk inhibitors: Design, synthesis,biological activity evaluation	Bioorganic & Medicinal Chemistry Letters	SCI
4	Energy-Transfer-Mediated Photocatalysis by a Bioinspired Organic Perylenephotosensitizer HiBRCP	Journal of Organic Chemistry	SCI
5	Progress in Synthesis and Bioactivity Evaluation of Pyrazoloquinazolines	Letters in Drug Design & Discovery	SCI
6	HPLC-ELSD法测定氨基酸原料药中5种糖类杂质	中国药科大学学报	CSCDC

2020年
序号	论文名称	来源期刊	收录情况
1	Emodin as a novel organic photocatalyst for selective oxidation of sulfides under mild conditions	RSC Advances	SCI
2	高效液相色谱-串联质谱法测定小鼠组织中的新型抗心力衰竭化合物AF-HF001	分析试验室	CSCDC
3	Synthesis and biological evaluation of diaryl urea derivatives as FLT3 inhibitors	Bioorganic & Medicinal Chemistry Letters	SCI
4	EGFR 抑制剂 AZD3759的合成工艺改进	中国药物化学杂志	CSCDE
5	奎扎替尼的合成	中国医药工业杂志	CSCDE
6	抗肿瘤药物恩曲替尼的合成工艺优化	化学试剂	统计源期刊
7	多靶点酪氨酸激酶抑制剂Lenvatinib的合成工艺优化	化学试剂	统计源期刊
8	HS-SPME-GC-MS法同时测定沙棘酒中11种酯类香气成分	分析试验室	CSCDC
9	柱前衍生化高效液相色谱法分析氨基酸原料药中的4种还原糖类杂质	分析试验室	CSCDC

2019年
序号	论文名称	来源期刊	收录情况
1	Determination of an isonicotinylhydrazide derivative, a novel positive inotropic compound, in mouse plasma by LC–MS/MS and its application to a pharmacokinetics study	Journal of Pharmaceutical and Biomedical Analysis	SCI
2	气相色谱法测定奥希替尼中溶剂残留量	沈阳药科大学学报	CSCDE
3	新型正电荷标记试剂的反应优化及应用	广州化工	统计源期刊
4	Perylenequinonoid-Catalyzed[4+1]and[4+2]Annulations of Azoalkenes:Photocatalytic Access to 1,2,3-Thiadiazole/1,4,5,6-Tetrahydropyridazine Derivatives	JOURNAL OF ORGANIC CHEMISTRY	SCI
5	Perylenequinonoid-catalyzed photoredox activation for the direct arylation of (het)arenes with sunlight	Organic & Biomolecular Chemistry	SCI
6	Cercosporin-bioinspired selective photooxidation reactions under mild conditions	Green Chemistry	SCI
7	Cercosporin-bioinspired photoreductive activation of aryl halides under mild conditions	Journal of Catalysis	SCI
8	Visible-light photocatalytic aerobic oxidation of sulfides to sulfoxides with a perylene diimide photocatalyst	Organic & Biomolecular Chemistry	SCI
9	氨基糖苷类抗生素的研究进展	中国新药杂志	CSCDC
10	Discovery and biological evaluation of novel G protein‐coupled receptor 119 agonists for type 2 diabetes	Archiv Der Pharmazie	SCI
11	Design, synthesis and biological evaluation of 2-(4-(methylsulfonyl)phenyl)pyridine derivatives as GPR119 agonists	Chemical Biology & Drug Design	SCI
12	靶向 Trk 抗肿瘤药物 larotrectinib 的新合成方法	中国药物化学杂志	CSCDE
13	Design, synthesis, and evaluation of a series of novel phenylpropanoic acid derivatives agonists for the FFA1	Chemical Biology & Drug Design	SCI
14	Isoliquiritigenin‐induced vasodilation by activating large-conductance Ca2+‐activated K+ channels in mouse mesenteric arteries	CLINICAL AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY	SCI
15	Cercosporin-photocatalyzed sp3 (C–H) activation for the synthesis of pyrrolo[3,4-c]quinolones	Organic & Biomolecular Chemistry	SCI
16	Metal-Free Cercosporin-Photocatalyzed C-S Coupling for the Selective Synthesis of Aryl Sulfides under Mild Conditions	European Journal of Organic Chemistry	SCI

2018年
序号	论文名称	来源期刊	收录情况
1	Synthesis and SAR of 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivatives as potent and selective CDK4/6 inhibitors	European Journal of Medicinal Chemistry	SCI
2	Cu-Catalyzed carbamoylation versus amination of quinoline N-oxide with formamides	ORGANIC & BIOMOLECULAR CHEMISTRY	SCI
3	Synthesis and biological evaluation of novel 5,6-dihydropyrimido[4,5-f] quinazoline derivatives as potent CDK2 inhibitors	BIOORGANIC & MEDICINAL CHEMISTRY LETTERS	SCI
4	可见光催化的丙炔酸酯三氟乙基化反应合成香豆素类似物	有机化学	SCI
5	N,N-二甲基甲酰胺二烷基缩醛对含N-H 化合物的N-烷基化反应	有机化学	SCI
6	新型抗血吸虫杂环化合物UPLC⁃QTOF⁃MS分析方法的建立	中国血吸虫病防治杂志	CSCDC
7	气相色谱法同时测定大蒜精油保健品中6 种活性有机硫化物	分析试验室	CSCDC
8	钠-葡萄糖共转运蛋白2抑制剂的研究进展	华西药学杂志	CSCDE
9	CDKs抑制剂BMS-265246的合成研究	中国药物化学杂志	CSCDE
10	抗癌新药帕布昔利布的合成工艺改进	中国药物化学杂志	CSCDE
11	TBAI 催化氨基羰基化合物与吲哚化合物的芳香化	广州化工	统计源
12	可见光催化下三氟甲基酮的选择性合成	广州化工	统计源
13	新型抗心衰化合物的合成及稳定性研究	广州化工	统计源

2017年
序号	论文名称	来源期刊	收录情况
1	Gold-Oxazoline Complex-Catalyzed Cross-Dehydrogenative Coupling of Glycine Derivatives and Alkenes	Advanced Synthesis and Catalysis	SCI
2	Transition-Metal-Free Trifluoromethylation of Aldehyde Derivatives with Sodium Trifluoromethanesulfinate	JOURNAL OF ORGANIC CHEMISTRY	SCI
3	Characterization and crystal structure of a novel zearalenone hydrolase from Cladophialophora bantiana	ACTA CRYSTALLOGRAPHICA SECTION F-STRUCTURAL BIOLOGY COMMUNICATIONS	SCI
4	三氟甲基亚磺酸钠实现的三氟甲基化反应研究进展	有机化学	SCI
5	AF-HF001对正常大鼠离体心脏的正性肌力及心电作用	中国药科大学学报	CSCDC
6	与2型糖尿病相关的G蛋白偶联受体激动剂的研究进展	中国新药杂志	CSCDC
7	RP-HPLC-DAD法快速测定沙棘叶中6种黄酮成分	中国药科大学学报	CSCDC
8	CDK抑制剂PHA-848125的工艺优化	中国医药工业杂志	CSCDE
9	GPR119激动药MBX-2982的合成	中国医药工业杂志	CSCDE
10	沙棘叶黄酮提取工艺的单因素研究及其品类变化	广州化工	统计源
11	GPR40激动剂药效团模型的构建及验证	计算机与应用化学	统计源
12	多指标-正交试验优化沙棘叶和沙棘籽中黄酮的提取工艺	中国药房	统计源

2016年
序号	论文名称	来源期刊	收录情况
1	5d, a novel analogue of 3-n-butylphthalide, decreases NADPH oxidase activity through the positive regulation of CK2 after ischemia/reperfusion injury	ONCOTARGET	SCI
2	Oxadiazole-2-oxides may have other functional targets, in addition to SjTGR, through which they cause mortality in Schistosoma japonicum	PARASITES & VECTORS	SCI
3	Iron-catalyzed direct α-arylation of α-amino carbonyl compounds with indoles	Organic and Biomolecular Chemistry	SCI
4	Immobilizing of oxo-molybdenum complex on cross-linked copolymer and its catalytic activity for epoxidation reactions	CATALYSIS COMMUNICATIONS	SCI
5	Cross-talk between 5-hydroxytryptamine and substance P in the melanogensis and apoptosis of B16F10 melanoma cells	EUROPEAN JOURNAL OF PHARMACOLOGY	SCI
6	Interferon-gamma Attenuates 5-Hydroxytryptamine-Induced Melanogenesis in Primary Melanocyte	BIOLOGICAL & PHARMACEUTICAL BULLETIN	SCI
7	Interleukin 10 protects primary melanocyte by activation of Stat-3 and PI3K/Akt/NF-kappa B signaling pathways	CYTOKINE	SCI
8	Gene Expression Profiling of H9c2 Cells Subjected to H2O2-Induced Apoptosis with/without AF-HF001	BIOLOGICAL & PHARMACEUTICAL BULLETIN	SCI
9	首个针对治疗高危神经母细胞瘤的新药dinutuximab	中国新药杂志	CSCDE
10	钠-葡萄糖共转运体2抑制剂研究进展	中国新药杂志	CSCDE
11	Synthesis of Aromatic Amide Derivatives and Their Biological Evaluation against Protein Tyrosine Phosphatase 1B and Scr Homology-2 Domain Containing Protein Tyrosine Phosphatase-2	有机化学	SCI
12	Cross-talk between interferon-gamma and interleukin-18 in melanogenesis	Journal of Photochemistry & Photobiology, B: Biology	SCI
13	天然大蒜精油对人体的排铅作用	分析科学学报	CSCDC
14	MK-3102关键中间体的合成工艺改进	广州化工	其他
15	邻氯苯甘氨酸甲酯的绿色合成工艺研究	广州化工	其他

2015年
序号	论文名称	来源期刊	收录情况
1	Zebrafish as a New Model for Phenotype-based Screening of Positive Inotropic Agents	CHEMICAL BIOLOGY & DRUG DESIGN	SCI
2	TBAI-catalyzed synthesis of alpha-ketoamides via sp(3) C-H radical/radical cross-coupling and domino aerobic oxidation	TETRAHEDRON LETTERS	SCI
3	Rh(I)-catalyzed decarbonylation synthesis of carbazoles via C-N cleavage	TETRAHEDRON	SCI
4	Palladium-Catalyzed Heck-Type Coupling via C-N Cleavage	SYNLETT	SCI
5	An efficient one-pot, three-component synthesis of vinyl sulfones via iodide-catalyzed radical alkenylation	TETRAHEDRON	SCI
6	Palladium(II)-Catalyzed C-H Acylation with Arylglycine Derivatives	SYNLETT	SCI
7	王不留行提取物对H_(22)荷瘤小鼠的抗肿瘤作用研究	Journal of Chinese Medicinal Materials	CSCD
8	含糖结构的抗糖尿病螺环化合物研究进展	Chinese Journal New Drugs	CSCD
9	手性胺拆分法制备雷美替胺	Chinese Journal of Synthetic Chemistry	CSCD
10	Synthesis of novel 3-aryl-1-oxa-2,8-diazaspiro[4.5]dec-2-ene derivatives and their biological evaluation against PTP1B	Chem Biol Drug Des	SCI
11	Asymmetric Catalytic Carbon-Carbon Coupling Reactions via Cross-Dehydrogenative Coupling Reactions	CHINESE JOURNAL OF ORGANIC CHEMISTRY	SCI
12	Mo Schiff base-tungstate ionic hybrid with enhanced heterogeneouscatalytic activity for epoxidation reactions	Applied Catalysis A: General	EI
13	Calcitonin gene-related peptide cooperates with substance P to inhibit melanogenesis and induces apoptosis of B16F10 cells	cytokine	SCI
14	阿普司特的合成工艺研究	广州化工	统计源
15	匹伐他汀关键手性中间体的立体选择性合成	广州化工	统计源
16	新型心肌肌球蛋白激动剂CK－1827452的合成研究	广州化工	统计源
17	GPR40 激动剂的合成	广州化工	统计源
18	浅谈以唤醒使命感为目标的本科教学	当代教育实践与教学研究	统计源
19	药物合成反应课程教学改革研究	广州化工	统计源
20	浅谈药理教学改革	广州化工	统计源
2014年
序号	论文名称	来源期刊	收录情况
1	Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors	BIOORGANIC & MEDICINAL CHEMISTRY LETTERS	SCI
2	Synthesis and In Vivo Hepatoprotective Activity of Some Novel Andrographolide Derivatives	LETTERS IN DRUG DESIGN & DISCOVERY	SCI
3	1H-2,3-Dihydroperimidine Derivatives: A New Class of Potent Protein Tyrosine Phosphatase 1B Inhibitors	MOLECULES	SCI
4	Design, Synthesis, and Biological Evaluation of Andrographolide Derivatives as Potent Hepatoprotective Agents	chemical biological & drug design	SCI
5	Iron-Catalyzed Oxidative Phosphonation of α-sp 3-c-H Bonds of N-Aryl Tetrahydroisoquinolines with Air as Oxidant	CHINESE J ORG CHEM	SCI
6	高效液相色谱-串联质谱法测定兔血浆中吡喹酮浓度	分析试验室	CSCD
7	金催化的吲哚对α －氨基酮的Friedel － Crafts 烷基化反应	广州化工	其他
8	微波辅助法合成手性β －氨基酸	广州化工	其他
2013年
序号	论文名称	来源期刊	收录情况
1	基底细胞癌新型治疗药物 vismodegib	中国新药杂志	CSCD
2	治疗心力衰竭的新策略——心肌肌球蛋白激动剂	中国新药杂志	CSCD
3	寓教于研的药物化学课程教学改革研究	广州化工	统计源
4	Synthesis and SAR studies of Praziquantel derivatives with activity against Schistosoma japonicum	Molecules	SCI
5	1-甲基-1，2，3，4-四氢异喹啉衍生物的合成及抗日本血吸虫活性评价	有机化学	SCI
6	王不留行提取物的急性毒理学研究	广州化工	统计源
2012年
序号	论文名称	来源期刊	收录情况
1	Au(III)-catalyzed intermolecular amidation of benzylic C–H bonds	Organic &Biomolecular Chemistry	SCI
2	Gold-Catalyzed Direct Indolation of Tetrahydroisoquinolines	Chinese Journal of Chemistry	SCI
3	Bu4NAuCl4 催化的H2O2 氧化的sp3-C—H 键与sp3-C—H 键的交叉偶联反应	有机化学	SCI
4	金配合物催化的吲哚对a,b-不饱和酮的Friedel-Crafts烷基化反应	有机化学	SCI
5	金催化的C—C 偶联反应研究进展	有机化学	SCI
6	药物化学课程教学改革	药学教育	统计源
7	Synthesis and Antiviral Activity of Conformational Analogues of Leucamide A	Molecules	SCI
8	优化制药工程专业药理学实验内容，培养学生创新能力	广州化工	统计源

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日期：2023-02-16 作者: . 来源：生命科学与健康工程学院